“SKF 96365 and FF also both significantly reduced desensitisation and prolonged the deactivation kinetics of the receptors to GABA (1mM; P<0.05).”
“Using whole cell patch-clamp recording to record … that SKF 96365 (1-100 μM) and FF (… GABA responses of recombinant human α1β2γ2 GABA(A) receptor stably expressed in HEK293 cells with IC(50) … GABA at all concentrations used in a manner consistent with a non-competitive mode of action.”